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Cat. No. Product Name Target Signaling Pathways
T35332 THZ1 2HCl

THZ1二盐酸盐,THZ1 2HCl,THZ1 Dihydrochloride

CDK Cell Cycle/Checkpoint
THZ1 2HCl (THZ1 Dihydrochloride) 是一种选择性、共价和变构的 CDK7 抑制剂,IC50 为 3.2 nM。 THZ1 2HCl 对多种癌细胞系具有抗增殖作用。
T3664 THZ1

CDK7 inhibitor,THZ1 2HCl

CDK Cell Cycle/Checkpoint
THZ1 (CDK7 inhibitor) 是一种新型的选择性强效共价 CDK7 抑制剂。它还抑制CDK12和CDK13,并下调 MYC 表达。
T7296 THZ2

CDK7-IN-1

CDK Cell Cycle/Checkpoint
THZ2 (CDK7-IN-1) 是 THZ1 的类似物,是一种有效的选择性 CDK7 抑制剂 ,IC50值为 13.9 nM。它有治疗三阴性乳腺癌的潜力。
T39459 THZ-P1-2

THZ-P1-2

THZ-P1-2 is a novel, specific inhibitor of PI5P4K that effectively targets PI5P4Kα. With an IC 50 of 190 nM, THZ-P1-2 selectively inhibits PI5P4Kα by forming covalent bonds with cysteine residues located on a disordered loop present in PI5P4Kα/β/γ. This mechanism not only disrupts autophagy but also elevates TFEB signaling. Moreover, THZ-P1-2 exhibits potent anticancer effects in leukemia cell lines, making it a promising candidate for therapeutic applications.
T23458 THZ1 Hydrochloride (1604810-83-4 free base)

THZ1 Hydrochloride

Others Others
THZ1 is a covalent inhibitor of CDK7 (IC50: 3.2nM).
T10546 bio-THZ1

CDK Cell Cycle/Checkpoint
bio-THZ1 is a biotinylated version of THZ1. THZ1 is a selective and irreversibly covalent CDK7 inhibitor (IC50: 3.2 nM).
T13153 THZ1-R

CDK Cell Cycle/Checkpoint
THZ1-R displays diminished activity for CDK7 inhibition(Kd:142 nM).
T72512 THZ1 Hydrochloride

THZ1 Hydrochloride,一种有效、选择性的共价CDK7抑制剂,IC50值为3.2 nM。它同样针对相关激酶CDK12和CDK13具有抑制作用,并能下调MYC表达。

化合物

THZ1 2HCl
Cat.No: T35332
Synonym: THZ1二盐酸盐,THZ1 2HCl,THZ1 Dihydrochloride
Target: CDK
THZ1
Cat.No: T3664
Synonym: CDK7 inhibitor,THZ1 2HCl
Target: CDK
THZ2
Cat.No: T7296
Synonym: CDK7-IN-1
Target: CDK
THZ-P1-2
Cat.No: T39459
Synonym: THZ-P1-2
Target:
THZ1 Hydrochloride (1604810-83-4 free base)
Cat.No: T23458
Synonym: THZ1 Hydrochloride
Target: Others
bio-THZ1
Cat.No: T10546
Synonym:
Target: CDK
THZ1-R
Cat.No: T13153
Synonym:
Target: CDK
THZ1 Hydrochloride
Cat.No: T72512
Synonym:
Target:
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